Substance / Medication

Buprenorphine

Overview

Active Ingredient
buprenorphine
RxNorm CUI
1819

Indications

Buprenorphine transdermal system is indicated for the management of severe and persistent pain that requires an opioid analgesic and that cannot be adequately treated with alternative options, including immediate-release opioids. Limitations of Use Warnings and Precautions (5.1) [see] Because of the risks of addiction, abuse, misuse, overdose, and death, which can occur at any dosage or duration and persist over the course of therapy, reserve opioid analgesics, including buprenorphine transderma

Labeler: Rhodes Pharmaceuticals L.P.Updated: 2026-02-03T00:00:00.000ZFull label on DailyMed

Boxed Warning

FDA Black Box Warning

Addiction, Abuse, and Misuse Warnings and Precautions (5.1) [see] Because the use of buprenorphine transdermal system exposes patients and other users to the risks of opioid addiction, abuse, and misuse, which can lead to overdose and death, assess each patient's risk prior to prescribing and reasse

Contraindications

When this intervention should not be used

Buprenorphine transdermal system is contraindicated in patients with: Warnings and Precautions (5.2) [see] Significant respiratory depression Warnings and Precautions (5.10) [see] Acute or severe bronchial asthma in an unmonitored setting or in the absence of resuscitative equipment Warnings and Pre

Indications & Related Conditions

Conditions associated via SNOMED clinical relationships

Administration & Protocol

Dosing, route, and treatment protocol

Detailed dosage and administration information is available in the full FDA drug label.

View full prescribing information on DailyMed

Monitoring & Follow-Up

Biomarkers relevant to this intervention via related conditions

No monitoring biomarkers have been mapped yet. Biomarker-intervention linkages are derived through related conditions and will expand as the knowledge graph grows.

Clinical Trials

35 trials linked to this intervention

35
Total Trials
3
Recruiting
14
With Results

Research Evidence

Published studies and systematic reviews

Sort:
Buprenorphine versus full agonist opioids for acute postoperative pain management: a systematic review and meta-analysis of randomized controlled trials.
Hickey Thomas R, Costa Gabriel P A, Oliveira Debora et al. · Reg Anesth Pain Med · 2026
PMID: 39753290Meta-Analysis
Strategy for effective analgesia with intravenous buprenorphine in patients with acute postoperative pain.
Szczupak Mateusz, Kobak Jacek, Cimoszko-Zauliczna Maria et al. · BMC Anesthesiol · 2025
PMID: 40287644Meta-AnalysisFull text (PMC)
Effectiveness of long-acting buprenorphine - A systematic review.
McMaster John, Abeysundera Hesitha · Australas Psychiatry · 2025
PMID: 39470393Meta-Analysis
Initiating buprenorphine to treat opioid use disorder without prerequisite withdrawal: an updated systematic review.
Adams Kathleen K, Waters Kristin, Sobieraj Diana M · Addict Sci Clin Pract · 2025
PMID: 39980050Meta-AnalysisFull text (PMC)
Multi-ancestry genome-wide association meta-analysis of buprenorphine treatment response.
Davis Christal N, Khan Yousef, Crist Richard C et al. · Neuropsychopharmacology · 2025
PMID: 40328918Meta-AnalysisFull text (PMC)
Initiation of buprenorphine in the emergency department or emergency out-of-hospital setting: A mixed-methods systematic review.
Armour Richard, Nielsen Suzanne, Buxton Jane A et al. · Am J Emerg Med · 2025
PMID: 39577213Meta-Analysis
Buprenorphine-naloxone versus buprenorphine for opioid use disorder during pregnancy: A systematic review and meta-analysis.
de Lima Fernanda Ribeiro, Molino Gabriela Oliveira Gonçalves, Gallo Ruelas Mariano et al. · Drug Alcohol Depend · 2025
PMID: 40073807Meta-Analysis
Incidence of buprenorphine-precipitated opioid withdrawal in adults with opioid use disorder: A systematic review.
Gregory Caroline, Yadav Krishan, Linders Jordyn et al. · Addiction · 2025
PMID: 39322991Meta-Analysis
Buprenorphine and Opioid Use Disorder Training: Graduate Nursing Curricula Recommendations.
Meadows Lauren, Simonton Amanda, Rolin Donna · J Psychosoc Nurs Ment Health Serv · 2024
PMID: 38095850Meta-Analysis

Research data from MEDLINE/PubMed

Benefits & Expected Outcomes

Benefits, expected outcomes, efficacy data, and NNT (Number Needed to Treat) are pending physician authorship and evidence review.

Risks & Side Effects

Adverse reaction and safety data for this drug is sourced from the FDA-approved label.

View adverse reactions & drug interactions on DailyMed

Related Symptoms

Symptoms associated with conditions this intervention addresses

No related symptoms have been mapped yet. Symptom linkages are derived through associated conditions.

Alternatives & Comparisons

Alternative treatments, comparison data, and clinical decision support are pending physician authorship.

Medical Disclaimer

This information is for educational purposes only and does not constitute medical advice, diagnosis, or treatment. Always consult with a qualified healthcare provider regarding any medical condition or treatment plan.

Do not start, stop, or change any treatment without consulting your healthcare provider.

Quick Facts

Type
Substance / Medication
Fully Specified Name
Buprenorphine (substance)
SNOMED CT
387173000
UMLS CUI
C0006405
RxNorm CUI
1819
Labeler
Rhodes Pharmaceuticals L.P.

Clinical Data

This intervention maps to 1 entities in the Ltrl knowledge graph.

1
Conditions
0
Biomarkers
0
Specialists
0
Symptoms
35
Clinical Trials

Data is sourced from SNOMED CT, UMLS, and the Ltrl clinical knowledge graph. Content sections marked as pending require physician authorship. Consult a healthcare provider before starting any treatment.

Buprenorphine — Conditions, Biomarkers & Specialists | Ltrl | Healos