Substance / Medication

Febuxostat

Overview

Active Ingredient
febuxostat
RxNorm CUI
73689

Indications

Limitations of Use: Febuxostat tablets are xanthine oxidase (XO) inhibitor indicated for the chronic management of hyperuricemia in adult patients with gout who have an inadequate response to a maximally titrated dose of allopurinol, who are intolerant to allopurinol, or for whom treatment with allopurinol is not advisable.Febuxostat tablets are not recommended for the treatment of asymptomatic hyperuricemia.

Labeler: Novadoz Pharmaceuticals LLCUpdated: 2026-02-20T00:00:00.000ZFull label on DailyMed

Boxed Warning

FDA Black Box Warning

[ Gout patients with established cardiovascular (CV) disease treated with febuxostat had a higher rate of CV death compared to those treated with allopurinol in a CV outcomes study see Warnings and Precautions (5.1)]. see Indications and Usage (1)]. [ Consider the risks and benefits of febuxostat wh

Contraindications

When this intervention should not be used

7 [see Drug Interactions ()] Febuxostat is contraindicated in patients being treated with azathioprine or mercaptopurine.

Indications & Related Conditions

Conditions associated via SNOMED clinical relationships

Administration & Protocol

Dosing, route, and treatment protocol

Detailed dosage and administration information is available in the full FDA drug label.

View full prescribing information on DailyMed

Monitoring & Follow-Up

Biomarkers relevant to this intervention via related conditions

No monitoring biomarkers have been mapped yet. Biomarker-intervention linkages are derived through related conditions and will expand as the knowledge graph grows.

Clinical Trials

13 trials linked to this intervention

13
Total Trials
1
Recruiting
8
With Results

Research Evidence

Published studies and systematic reviews

Sort:
The efficacy and safety of different doses of febuxostat and allopurinol: A meta-analysis.
Zhang Feng, Wang Yanyan · Jt Dis Relat Surg · 2025
PMID: 40783988Meta-AnalysisFull text (PMC)
Cardiovascular Safety of Febuxostat in Patients With Gout or Hyperuricemia: A Systematic Review of Randomized Controlled Trials.
Ghossan Roba, Aitisha Tabesh Ouidade, Fayad Fouad et al. · J Clin Rheumatol · 2024
PMID: 38115182Meta-Analysis
Association between use of febuxostat and muscle injury: A disproportionality analysis and meta-analysis of randomized controlled trials.
Mitsuboshi Satoru, Kotake Kazumasa · Br J Clin Pharmacol · 2023
PMID: 36585759Meta-Analysis

Research data from MEDLINE/PubMed

Benefits & Expected Outcomes

Benefits, expected outcomes, efficacy data, and NNT (Number Needed to Treat) are pending physician authorship and evidence review.

Risks & Side Effects

Adverse reaction and safety data for this drug is sourced from the FDA-approved label.

View adverse reactions & drug interactions on DailyMed

Related Symptoms

Symptoms associated with conditions this intervention addresses

No related symptoms have been mapped yet. Symptom linkages are derived through associated conditions.

Alternatives & Comparisons

Alternative treatments, comparison data, and clinical decision support are pending physician authorship.

Medical Disclaimer

This information is for educational purposes only and does not constitute medical advice, diagnosis, or treatment. Always consult with a qualified healthcare provider regarding any medical condition or treatment plan.

Do not start, stop, or change any treatment without consulting your healthcare provider.

Quick Facts

Type
Substance / Medication
Fully Specified Name
Febuxostat (substance)
SNOMED CT
441743008
UMLS CUI
C0249529
RxNorm CUI
73689
Labeler
Novadoz Pharmaceuticals LLC

Clinical Data

This intervention maps to 1 entities in the Ltrl knowledge graph.

1
Conditions
0
Biomarkers
0
Specialists
0
Symptoms
13
Clinical Trials

Data is sourced from SNOMED CT, UMLS, and the Ltrl clinical knowledge graph. Content sections marked as pending require physician authorship. Consult a healthcare provider before starting any treatment.