Substance / Medication

Gefitinib

Overview

Active Ingredient
gefitinib
RxNorm CUI
328134

Indications

Clinical Studies (14) see Gefitinib tablets are indicated for the first-line treatment of patients with metastatic non-small cell lung cancer (NSCLC) whose tumors have epidermal growth factor receptor (EGFR) exon 19 deletions or exon 21 (L858R) substitution mutations as detected by an FDA-approved test []. Clinical Studies (14) see Limitation of Use: Safety and efficacy of gefitinib tablets have not been established in patients with metastatic NSCLC whose tumors have EGFR mutations other than ex

Labeler: Ingenus Pharmaceuticals, LLCUpdated: 2023-12-28T00:00:00.000ZFull label on DailyMed

Contraindications

When this intervention should not be used

None.

Indications & Related Conditions

Conditions associated via SNOMED clinical relationships

Administration & Protocol

Dosing, route, and treatment protocol

Detailed dosage and administration information is available in the full FDA drug label.

View full prescribing information on DailyMed

Monitoring & Follow-Up

Biomarkers relevant to this intervention via related conditions

No monitoring biomarkers have been mapped yet. Biomarker-intervention linkages are derived through related conditions and will expand as the knowledge graph grows.

Clinical Trials

3 trials linked to this intervention

3
Total Trials
0
Recruiting
3
With Results

Research Evidence

Published studies and systematic reviews

Sort:
Genetic Variants in theandGene Drug Transporters Involved in Gefitinib-Associated Adverse Reaction: A Systematic Review and Meta-Analysis.
Morau Mariana Vieira, Seguin Cecília Souto, Visacri Marília Berlofa et al. · Genes (Basel) · 2024
PMID: 38790220Meta-AnalysisFull text (PMC)
Impact of ABCG2 rs2231142(421C>A) Variant on the Clinical Outcomes of Patients With-mutated Non-small Cell Lung Cancer Treated With Gefitinib: A Comprehensive Meta-analysis.
DE Moraes Francisco Cezar Aquino, Souza Maria Eduarda Cavalcanti, DA Silva Emanuele Rocha et al. · Anticancer Res · 2024
PMID: 39626927Meta-Analysis
The efficacy of gefitinib supplementation for breast cancer: A meta-analysis of randomized controlled studies.
Ye Jing, Tian Tian, Chen Xiaopin · Medicine (Baltimore) · 2020
PMID: 33120749Meta-AnalysisFull text (PMC)
A meta-analysis of the safety and effectiveness of pemetrexed compared with gefitinib for pre-treated advanced or metastatic NSCLC.
Lu Xiaoxin, Li Shengshu, Chen Weizong et al. · Medicine (Baltimore) · 2020
PMID: 32702875Meta-AnalysisFull text (PMC)
Gefitinib provides similar effectiveness and improved safety than erlotinib for advanced non-small cell lung cancer: A meta-analysis.
Zhang Wenxiong, Wei Yiping, Yu Dongliang et al. · Medicine (Baltimore) · 2018
PMID: 29668619Meta-AnalysisFull text (PMC)
Gefitinib for advanced non-small cell lung cancer.
Sim Esther Ha, Yang Ian A, Wood-Baker Richard et al. · Cochrane Database Syst Rev · 2018
PMID: 29336009Meta-AnalysisFull text (PMC)

Research data from MEDLINE/PubMed

Benefits & Expected Outcomes

Benefits, expected outcomes, efficacy data, and NNT (Number Needed to Treat) are pending physician authorship and evidence review.

Risks & Side Effects

Adverse reaction and safety data for this drug is sourced from the FDA-approved label.

View adverse reactions & drug interactions on DailyMed

Related Symptoms

Symptoms associated with conditions this intervention addresses

No related symptoms have been mapped yet. Symptom linkages are derived through associated conditions.

Alternatives & Comparisons

Alternative treatments, comparison data, and clinical decision support are pending physician authorship.

Medical Disclaimer

This information is for educational purposes only and does not constitute medical advice, diagnosis, or treatment. Always consult with a qualified healthcare provider regarding any medical condition or treatment plan.

Do not start, stop, or change any treatment without consulting your healthcare provider.

Quick Facts

Type
Substance / Medication
Fully Specified Name
Gefitinib (substance)
SNOMED CT
407100002
UMLS CUI
C1122962
RxNorm CUI
328134
Labeler
Ingenus Pharmaceuticals, LLC

Clinical Data

This intervention maps to 1 entities in the Ltrl knowledge graph.

1
Conditions
0
Biomarkers
0
Specialists
0
Symptoms
3
Clinical Trials

Data is sourced from SNOMED CT, UMLS, and the Ltrl clinical knowledge graph. Content sections marked as pending require physician authorship. Consult a healthcare provider before starting any treatment.